I-Heptral yipropati enefuthe le-hepatoprotective, efumaneka kwiindlela ezimbini: iipilisi zomlomo kunye nama-ampoule ukuphathwa kwe-intravenous okanye ye-intramuscular. I-Medication Heptral kwi-ampoules yi-lyophilizate (powder) yokulungiselela isisombululo esinikezelwa ngayo isisombululo esisodwa.
Isithako esisebenzayo sesilwayo yi-ademethionine, into ephilayo equlethwe kuzo zonke izicubu zomzimba. Idlala indima ebalulekileyo kwiinkqubo ezininzi zezinto eziphilayo kwaye ikhuthaza ukwanda kwindlela yokukhusela yamaseli esebindi. Ukubunjwa kwe-solvent kufaka izinto ezifana nale:
- I-l-lysine (i-amino acid);
- hydroxyde
- amanzi o lu ngiweyo.
Impembelelo ye-Pharmacological yeenjini kunye neHeptral
Isenzo salo mfuziselo sijoliswe, okokuqala, ekubuyiselweni kweenkqubo zeethambo ezinqamlekileyo kwiiseli ze-hepatic kunye nokuhlaziywa kwezicubu. Kodwa, ngaphezu koko, i-heptral inefuthe elihle kwimisebenzi yengqondo.
Unyango lwe-Heptral njengesisombululo sokufakelwa ijokelelo kunceda oku kulandelayo:
- ukuveliswa kwe-bile acid production;
- ukuphuculwa kwe-motility yesigca esiswini;
- ukuzaliswa kwe-admetionin ukulahleka emzimbeni kunye nokusebenza komveliso wayo;
- ukukhuselwa kweeseli zesibindi ukusuka kwiibhokhwe;
- isithintelo sokwandiswa kwezicubu ezinxulumene nesibindi;
- ukuphuculwa kokuqhutyelwa kweengxaki zentliziyo;
- ukuqhutyelwa kwenkqubo yesistim ephakathi, njl
Izibonakaliso zokutyunjwa kwe-heptral kwi-ampoules
Iinjongo ze-Heptral zicetyiswa ukuba zithwale izifo:
- i-hepatitis engapheliyo;
- i-hepatosis ;
- cholecystitis engapheliyo;
- cholestasis intrahepatic;
- i-cirrhosis yesibindi;
- cholangitis ;
- umonakalo wesibindi sesimo esiyingozi (i-viral, utywala, iziyobisi, njl.);
- umonakalo wengqondo;
- i-abstinence syndrome (i-narcotic, utywala, njl njl);
- ukuxinezeleka.
Ukungqinelana nokusetyenziswa kwe-heptral
Ngokwemiyalelo, i-Heptral kwi-ampoules ayimisiwe kwiimeko ezilandelayo:
- ukukhulelwa (I - II trimesters);
- ixesha lokuncelisa;
- ukunyanzelwana komntu kumacandelo esilwayo;
- ukusilela kwe-cystathione-beta synthase;
- ingxaki yokuxilongwa kwe-cyanocobalamin.
Qaphela, le nkunkuma imiselwe ukuhluleka komntu, kunye neengxaki ze-bipolar, kwakunye nezigulane ezigugile.