UValsartan ubhekisela kwiziyobisi ezingekho emlonyeni onomhlaba onqanda ama-receptors ye-angiotensin II. Kwiminyaka eyisixhenxe elandelelanayo, ukususela ngo-2008, iyeza liye laziwa njengezilwanyana ezithandwayo kakhulu kwihlabathi ukuze unyango lwe-hypertension.
Inzuzo yeValsartan kukuba ayiyikuvimbela i-enzyme yokuguqula i-angiotensin, oko kukuthi, iikhemikhali zendalo kunye nezomculo. UValsartan wenza ngenye indlela, oko kutheni kubonwa. Ukongezelela, ayivimbeli i-receptors yama-hormone okanye iziteshi ze-ion, ezibalulekileyo ekuqhelweni komsebenzi wenkqubo ye-cardiovascular system. Ukufaneleka kwesi sidakamizwa kubandakanya ukungabikho kwesiphumo esibi kwizinga le- cholesterol epheleleyo, i-glucose kunye ne-uric acid kwi-plasma.
Ukubunjwa kwe-Valsartan yokulungiselela
Isithako esisebenzayo sokulungiselela i-valsartan, njengezinto ezincedisayo:
- i-magnesium stearate okanye i-acaric acid-isakhi setyuwa, i-magnesium kunye ne-acaric acid, ebonakalayo yendalo yamachiza;
- MCC (i-microcrystalline cellulose), eyenzelwe ukucoca i-membrane yamathumbu emathumbu amancinci;
- I-Croscarmellose - i-sodium ityuwa ye-cellulose inomsebenzi obalulekileyo (unceda ukutshabalalisa iziyobisi emathunjini);
- i-aerosil - i-thickener ne-sorbent;
- idayi "Opadrai Pink".
Uninzi lwezityalo zeValsartan alusebenzi kwimveliso yezobisi, kubangelwa ukusebenza kwezinto eziphambili. Kukho izidakamizwa ezidibeneyo iValsartan + i-hydrochlorothiazide, equka i-hydrochlorothiazide into engavimba ukubuyisela kwakhona i-sodium, i-chlorine kunye ne-ion yamanzi.
Ungathatha njani uValtrasan?
Njengoko umyalelo wokusetyenziswa kweziyobisi uValsartan uthi, le nyeza ithathwa ngomlomo. Kule nkqubo yenziwa kabini ngemini ibe ngu-40 mg yesilwanyana, okanye kanye, kodwa i-80 mg. Ukuba isiphumo esilindelekileyo asifezekanga ngexesha elimiselweyo, umthamo ungancipha ngokuthe ngcembe, ngelixa kuphela ugqirha angayilungisa le nto. Ukuzinyango kwimeko enokuyenza ingozi enkulu.
Ndingayinceda njani uValsartan?
Iyezabisi zeValsartan zinenani elifanayo, phakathi kwazo:
- Ukukhupha;
- Corinfar;
- Sakur;
- Cardura;
- Tonusin.
Into esebenzayo ye- Enap iyona enalapril, eneendawo ezifanayo kwi-valsartan, ngoko ke izibonakaliso zokusetyenziswa kweziyobisi ziyafana: ukuxinzeleleka komfutho wegazi kunye nokuhluleka kwentliziyo.
I-Corinfar ijoliswe ekunyangeni izifo zeentliziyo ezahlukeneyo, ngoko kukho izikhombisi ezininzi zokusetyenziswa kwayo. Into esebenzayo yeziyobisi yi-nifedipine, eyaziwa nge-calcium channel blocker. Kodwa, ngelishwa, eli liyeza linoluhlu olude lweempembelelo, ezibandakanya iingxaki ngesondlo sesisu, isibindi, isistim se-cardiovascular system kunye ne-hematopoiesis system, kunye neempembelelo zokugula.
I-Sakur inesicelo esincinci - unyango lwexinzelelo lwengcinezelo, ngoko ke i-analogue ethandwa kakhulu yiValsartan. Ngokuqhelekileyo, isilwanyana sisetyenziswa ngokubambisana nezinye iziyobisi. Inkunkuma esebenzayo i-Sakura yi-lacidippin - i-blocker yeziteshi ze-calcium ezicothayo.
Isidakamizwa i-Kardura sisetyenziswe njengeyeza lokuqala kumachiza kunyango lwe-hypertension kunye nomsebenzi walo oyintloko kukulawula uxinzelelo lwegazi. Into esebenzayo yi doxazosin, ephikisanayo kwizigulane ezine-hypersensitivity kuphela. Uluhlu olude lweempembelelo kwimimiselo yokusetyenziswa kwesi sifaniso seValsartan nawe awuyi kufumana, ngoko ke izidakamizwa iKardura zinokuthi zithathwe njengomncintiswano ofanelekileyo weValtrasan.
I-Tonusin isekelwe kwizixhobo zezityalo kwaye iyakwazi ukuba nefuthe eliyinkimbinkimbi, ngoko isetyenziswe njenge-toning jikelele, i-normalizing blood pressure, indlela yokubuyisela. I-Tonusin iphinda isetyenziswe njengeliyeza elithuthukisa ukujikelezwa kwe-coronary kunye ne-peripheral circulation kunye nefuthe le-cardiac output.