Ukulwa nezifo ezifayilini, izidakamizwa ezininzi ziveliswa namhlanje. Kwaye phambi kokuba ugqirha kukho ukhetho olunzima lweyeza eliphezulu kakhulu kule ndawo okanye kwimeko.
Amacwecwe e-Ketoconazole okanye amanye amalungiselelo esekelwe kuwo angama-agent antifungal of action wide. Banceda ukunyanga i-mycoses yenkqubo, oko kukuthi, izifo ezibangelwa yi-fungi, kunye nezifo ezifakwe kwi-fungal - i-mycoses, i-seborrhea.
I-Ketoconazole inomphumo onobungozi kwi-fungus-like fungus ye-genus Candida, i-dermatophytes, i-mold fungus, i-pathogens eyahlukeneyo ye-mycoses yesistimu kunye ne-staphylococci kunye ne-streptococci.
Iipilisi zeCetoconazole zichazwe nini?
Izimpawu zokusetyenziswa kwe-ketoconazole zi:
- ukusuleleka kwefungal of tractes tract;
- izifo ezithinta izifo zomzimba, okubandakanya i-candidiasis yesisu, eyaziwa ngokuba yi-thrush, kunye ne-candidiasis engamaqabane;
- i-mycosis yezikhonkwane, isikhumba, iinwele, i-paronychia, i-folliculitis;
- i-seborrheic dermatitis (dandruff);
- septicemia ekhunjini;
- iliso le-mycosis;
- i-mycoses ye-systemic - candidiasis, blastomycosis, i-histoplasmosis, njl.;
- ukuthintela ukusuleleka kwezifayilini kubantu abane-immunodeficiency kunye neengozi yokwanda kwezilonda zefungal.
Xa uthathwa ngomlomo, amalungiselelo kwiipilisi kunye ne ketoconazole anika unyango osebenzayo kwi-surface and systemic mycoses. Isenzo salo nxu lumene nokutshatyalaliswa kwenkqubo ye-biosynthesis ye-ergosterol phospholipids kunye ne-triglycerides, echaphazelekayo ekubunjweni kwesikhumba sefenal. Ekugqibeleni, ukukhula nokuphindaphinda kwala maseli anobungozi kuyaphela kwaye isifo sifana.
Xa kuthathwa ngomlomo, ukulungiswa ngokucokisekileyo, oko kukuthi, kungena kwigazi, kusasazeka kwiifom, inxalenye encinci ingene kwi-cerebrospinal fluid. Emva kokungena kwi-digestive tract, i-active active is metabolized in the liver, yakha inani elikhulu leemetabolites ezingasebenzi. Isilwanyana sidityaniswe kumchamo (13%), sidityaniswe ne-bile kwaye sidityaniswe ngamanzi (57%).
Ngokuqhelekileyo iipilisi 1-2 zithathwa ngosuku kunye nokutya kweeveki ezi-2-8, kuxhomekeke kwisifo kunye nesisindo somzimba. Isiza lingalawulwa kwabantwana abangaphezu kweminyaka eyi-12 ubudala.
Ukuchasana kunye nemiphumo emibi ngokuthatha iKetoconazole
Amacwecwe e-Ketoconazole avela kwi-seborrheic dermatitis kunye nezinye izifo ze-etymology ye-fungal zichazwe ngokukhulelwa, ngononophelo, abantwana abaneminyaka engaphantsi kwe-12 ubudala, abantu abane-hypersensitivity ketoconazole kunye nokuphazamiseka okukhulu kwe-kidney kunye nesibindi somsebenzi.
Iziphumo ezichaphazelekayo zokuthatha amacwecwe zilandelayo:
- isicaphulo kunye nokuhlanza;
- isifo sohudo;
- ingxaki yokulala;
- utywala, intloko;
- ukulahlekelwa kweenwele;
- paresthesia;
- exanthema;
- kunciphisa umnqweno wesini;
- gynecomastia;
- urticaria, ukugqithisa kwesikhumba;
- photophobia;
- umkhuhlane.
Ukulawulwa komlomo kwamalungiselelo asekelwe kwi-ketoconazole kufuneka kuhambisane nokulawulwa kwonyango rhoqo: ukuhlolwa kwegazi, ukukhangela isibindi kunye nemisebenzi yengqondo. Ukungathandabuzeki ngokucacileyo ekuzijoliseni nasekuziphatheni ngamachiza ngamachiza. Unyango lunokumiselwa kuphela ngugqirha.
Kwimeko ye-fungal meningitis, ukusetyenziswa kwe-ketoconazole akucebisi, kuba loo nto ingenanga kakuhle nge-BBB (umqobo we-hemato-encephalic).
Ukulungiselelwa okusekelwe kule nkunkuma yi-hepatotoxic, ngoko ke kufuneka isetyenziswe kuphela xa inzuzo enokuthi ibhekise umngcipheko. Ngokukodwa kubangelwa ngaba gulane abanomsebenzi ophezulu ngokwemvelo ye-enzyme okanye ewonakalisa umonakalo kwisibindi ngenxa yokuthatha ezinye iziyobisi.
Ukulungiselela nge ketoconazole kwiipilisi
Nantsi amagama eengqungquthela zesakhiwo se ketoconazole kwiipilisi (ngokubhekiselele kwisithako esisebenzayo):
- Mycosorrhal;
- Fungistab;
- Dermazol;
- Oronazole;
- INizoral ;
- KetoconazoleAltapharm;
- Ketoconazole DS;
- Mikanisal;
- Livarol;
- Mikoket;
- Fungin.