Desloratadine kunye ne-loratadine --hluko

Ukuze uqonde ngokukhawuleza into efunayo, khumbula isilwanyana esithandwayo njengoErius . Le yindlela eqhelekileyo yokulungisa unyango. Isithako sayo esisebenzayo, i-desloratadine, i-metabolite ye-loratadine. Le nto yabangela iziphumo ezahlukeneyo zezinto ezimbini. Desloratadine kunye ne-loratadine, ulwahlulo lwalo luboniswe ngezantsi, ngokukhawuleza ukulwa nokuxhomekeka kweengxaki ezihlukahlukeneyo, ukukhulula ubuqhophololo kwaye usebenzise isenzo sokuchasana.

Uwuphi umehluko phakathi kwe-loratadine kunye ne-desloratadine?

Zombini izinto ezivimba i-histamine n1 receptors. Abenayo isenzo se-cardiotoxic kunye ne-hypnotic, basuswa ngokukhawuleza emzimbeni ngaphandle kokulibala.

Nangona kunjalo, i-desloratadine yi-loratadine metabolite, oko kukuthi, ngumveliso wokwenziwa. Ngaloo ndlela, xa ethatha i-loratadine, yena, ngaphambi kokuba aqalise isenzo sakhe, iya kuba yinto yokuhlambalaza. Ngenxa yoko, oku kuhamba ngokukhawuleza kunokuba kulungiselelwe isizukulwana esidlulileyo, kuba akudingeki ukuba iguqulwe kwisitya sokugqibela.

Yiyiphi enye ingcono - desloratadine okanye i-loratadine?

Iintlobo ze-desloratadine ziquka ukusebenza kwayo. Kuyixesha eli-4-15 elisebenza ngakumbi kunokuba lidlulileyo. Oku kuvumela ngokukhawuleza kufinyelele ingqwalaselo ephezulu kunye nokunciphisa umlinganiselo kwisigamu.

Kubalulekile ukuba uqaphele ukuba ezininzi iziyobisi ezisekelwe kwi-desloratadine zithengiswa njenge-siraphu, okwenza kube lula ukuphatha abantwana, ukuqala ngeenyanga ezintandathu.

Ukuqwalasela i-desloratadine kunye ne-loratadine kwaye uphendule lo mbuzo yintoni umehluko, kuyafaneleka ukuba uqaphele ukuba xa kufuneka okokugqibela, ukusebenza ngokuqhelekileyo kwesibindi kuyadingeka. Emva koko, kwimeko yonyango, ukuguqulwa kwi-desloratadine kuya kuba nzima.

Iindleko zeziyobisi ezisekelwe kwi-desloratadine ngumyalelo wobukhulu obuphezulu kunelo loratadine. Iyeza lokugqibela kufuneka linikezelwe ngokukhethekileyo ukuba kuyimfuneko ukulwa namaxesha angatshatyalaliswayo, ngokungabikho kwezifo zesibindi.