Anaprilin analogues

I-Anaprilin yisilwanyana esivela kwiqela le-beta-blockers ebonisa i-antianginal, hypotensive kunye ne-antiarrhym properties. Le yonyango elisebenzayo, elithengiyo kwaye elingabizi elinokukhawuleza ukunciphisa izinga lentliziyo kunye noxinzelelo lwegazi, ukuphelisa ukuhlaselwa kwe-panic, kunye nokunciphisa imeko kwezinye izifo. Nangona kunjalo, eli liyeza alinakho imiphumo emibi kwaye lingasetyenziselwa kuphela phantsi kweliso logqirha, kwaye kwezinye iimeko zichazwe ngokusetyenziswa. Ngaba zifana neAnadrilin ngaphandle kwemiphumo emibi, kwaye yintoni ukuphumelela kwayo, siya kuqwalasela.


Iintetho zeAnaprilin

Isilwanyana esixutyushwa njengesiqhelo esisebenzayo esinezixhobo eziqukethe ipropranolol hydrochloride. Izifaniso zesakhiwo (izifaniso) zeAnaprilin, eziqukethe into efanayo esebenzayo, ngamachiza alandelayo:

Ekubeni iimveliso ezidwelisweyo zifana nokubunjwa, ngoko ke, ngokwemiqondiso, ukuchasiswa kunye nemiphumo emibi, ziyakutshintshana.

Kukho izifaniso ze-Anaprilin kungekhona ngokutsho kwezinto ezisebenzayo, Ezi ziyizidakamizwa zeqela le-pharmacological (beta-blockers) kunye nokubonisa iimpawu ezifanayo, kodwa kubandakanye nezinye izinto ezisebenzayo. Ukongezelela, namhlanje kukho iziyobisi ezikhuselekileyo ezineendlela ezifanayo zokuthatha isenzo - ezikhethiweyo (ezikhethiweyo) beta-blockers. Ezi zi yobisi, ngokungafani ne-Anaprilin engakhethiyo, vimba umsebenzi wezinto ezithile kuphela zee-organes ze-beta-adrenergic receptor, ezifunekayo ukuba zenze. Ngaloo ndlela, akukho miphumo kwezinye iimbumba, kwaye inani lemiphumo engafanelekanga kwonyango olunjalo lonyango luyancitshiswa kakhulu.

Ezi zifana zanamhlanje zakwaAnaprilin ngamachiza alandelayo:

Ukulungiswa kwoluhlu olukhankanywe ngasentla luhluke ekuhlaleni kwabo, ubude bentshukumo, ixesha lokunyusa kunye nezinye izikhombisi. Isigqibo sokuba zezi zonyango kufuneka zisetyenziswe unyango zingathathwa kuphela ngugqirha ngokwazo, ngokusekelwe kwidatha yezifundo zokuxilonga, iimpawu zesigulane somzimba kunye nokunyamezela kwamachiza.

Kunokuba kunokwenzeka ukuthatha indawo ye-Anaprilin kwi-tachycardia kwi-thyrotoxicosis?

I-Thyrotoxicosis yimeko ebangelwa yintsholongwane ye-hormone ye-thyroid, apho zonke iinkqubo ze-metabolic emzimbeni zikhawuleza. Izigulane ezinokuxilongwa rhoqo, nangona zilala, zixhala malunga nokukhula kwenhliziyo - tachycardia. Isidingo somzimba we-cardiac in oxygen sanda, umzimba usebenza ngokugqithisa. Ukongeza, kwizigulane ezine-thyrotoxicosis zenzeka ukuhlaselwa kwesiphazamiso senhliziyo (kubandakanywa i-fibrillation ye-atrial), i-angina pectoris.

Ngaloo sifo, i-tachycardia ayinakunqandwa nakwixesha lokusebenzisa iziyobisi ezithintelayo kwezinye iimeko - i-cardiac glycosides (ngaphandle kokuba isetyenziswe ngaphandle kweziyobisi ezinciphisa imveliso ye-hormone ye-thyroid). Ngokukhawuleza ukuphucula imeko yesigulane kwimeko enjalo iAnaprilin (kunye nezinye iziyobisi ezisekelwe kwipropranolol), nto leyo eyanciphisa izinga le-hormone ye-thyroid. Ngokumalunga neempawu zeAnaprilin, ezinxulumene ne-beta-blockers ekhethiweyo, impembelelo yabo kwi-tachycardia ngenxa ye-thyrotoxicosis ayisebenzisekanga. le mali ayinciphisi izinga le-T3.